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Search Results for " imidazoline receptor "

20

Compounds

Cat No. Product Name Synonyms Targets
T22051 BU 224 hydrochloride Imidazoline Receptor
BU 224 hydrochloride is a selective imidazoline I(2) binding site ligand and has antinociceptive and antidepressant-like activities.
T6641 Rilmenidine Phosphate Apoptosis , Adrenergic Receptor , Autophagy , Imidazoline Receptor
Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.
T3158 Harmane Loturine,Harman,Aribine Adrenergic Receptor , Monoamine Oxidase , Imidazoline Receptor
Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.
T0115 Idazoxan hydrochloride RX 781094 Adrenergic Receptor , Imidazoline Receptor
Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.
T0925 Allantoin Glyoxyldiureide,5-Ureidohydantoin Endogenous Metabolite , Imidazoline Receptor
Allantoin (Glyoxyldiureide), a urea hydantoin found in urine and plants, is used in dermatological preparations.
T22052 BU 226 hydrochloride Imidazoline Receptor
BU 226 hydrochloride demonstrates affinity for imidazoline (I) receptors, in particular the I2 binding site with a Ki of 1.4 nM. BU 226 hydrochloride showed low (microM) affinity for alpha 2-adrenoceptors.
T1028 Moxonidine BDF5895 Imidazoline Receptor
Moxonidine (BDF5895) is a selective agonist at the imidazoline receptor subtype 1, acting as an antihypertensive drug.
T4808 Agmatine sulfate Agmatine sulfate salt Endogenous Metabolite , NO Synthase , Imidazoline Receptor
Agmatine sulfate (Agmatine sulfate salt) is a bioactive metabolite of the arginine amino acid. It exerts modulatory action at multiple molecular targets, such as neurotransmitter systems, ion channels and nitric oxide sy...
T23283 2-Methoxyidazoxan monohydrochloride RX 821002 hydrochloride Adrenergic Receptor
L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor, with little or no antagonistic effect on imidazoline. It has a significantly higher affinity ...
T15010 CR4056 6-(1H-imidazol-1-yl)-2-phenylquinazoline MAO , Imidazoline Receptor
CR4056 (6-(1H-imidazol-1-yl)-2-phenylquinazoline) is a selective inhibitor of MAO-A with IC50 of 202.7 nM and a ligand of I2-imidazoline receptor with IC50 of 596 nM.
T6703 Tetrahydrozoline hydrochloride Murine Plus,Tetryzoline hydrochloride,Tyzine,Tetrahydrozoline HCl Adrenergic Receptor
Tetrahydrozoline hydrochloride (Murine Plus) is an imidazoline derivative with alpha receptor agonist activity.
T22492 2-BFI hydrochloride Imidazoline Receptor
2-BFI hydrochloride is a high-affinity agonist of I2-imidazoline receptor. 2-BFI hydrochloride can be used in studies about protection against stroke and acute inflammatory immune disease.
T21911 Rilmenidine hemifumarate Rilmenidine (hemifumarate),S-3341 hemifumarate Apoptosis , Imidazoline Receptor
Rilmenidine hemifumarate (S-3341 hemifumarate) is a novel, orally active and selective I1 imidazoline receptor and α2-adrenoceptor agonist that induces autophagy, regulates the proliferation of leukaemia cells, stimulate...
T23263 RS 45041-190 hydrochloride Others
Highly selective I2 imidazoline receptor ligand
T22760 Efaroxan hydrochloride Others
α2 adrenoceptor antagonist and imidazoline I1 receptor ligand
T26171 S23757 S-23757,S 23757
S23757 is an imidazoline 1 receptor (I1R) selective ligand.
T68931 Tracizoline
Tracizoline is a potent I2-imidazoline receptor agonist.
T40869 Moxonidine hydrochloride BDF5895hydrochloride
Moxonidine Hydrochloride serves as a selective agonist for the imidazoline receptor subtype 1 and functions as an antihypertensive agent. It primarily acts within the central nervous system and demonstrates a significant...
T27155 Dexisometheptene TNX 201,TNX-201,(R)-Isometheptene,TNX201
Dexisometheptene is an antimigraine drug candidate. Dexisometheptene significantly increases the pain threshold of acute pain response, and potently and selectively binds to receptors in the central nervous system known ...
T73214 RX 801077 2 BFI free base
RX 801077 (2 BFI free base), a selective imidazoline I2 receptor (I2R) agonist, exhibits a K i value of 70.1 nM, demonstrating anti-inflammatory and neuroprotective properties. This compound holds research potential for ...

Compounds

BU 224 hydrochloride
T22051
Synonym:
Target: Imidazoline Receptor
Rilmenidine Phosphate
T6641
Synonym:
Target: Apoptosis, Adrenergic Receptor, Autophagy, Imidazoline Receptor
Harmane
T3158
Synonym: Loturine,Harman,Aribine
Target: Adrenergic Receptor, Monoamine Oxidase, Imidazoline Receptor
Idazoxan hydrochloride
T0115
Synonym: RX 781094
Target: Adrenergic Receptor, Imidazoline Receptor
Allantoin
T0925
Synonym: Glyoxyldiureide,5-Ureidohydantoin
Target: Endogenous Metabolite, Imidazoline Receptor
BU 226 hydrochloride
T22052
Synonym:
Target: Imidazoline Receptor
Moxonidine
T1028
Synonym: BDF5895
Target: Imidazoline Receptor
Agmatine sulfate
T4808
Synonym: Agmatine sulfate salt
Target: Endogenous Metabolite, NO Synthase, Imidazoline Receptor
2-Methoxyidazoxan monohydrochloride
T23283
Synonym: RX 821002 hydrochloride
Target: Adrenergic Receptor
CR4056
T15010
Synonym: 6-(1H-imidazol-1-yl)-2-phenylquinazoline
Target: MAO, Imidazoline Receptor
Tetrahydrozoline hydrochloride
T6703
Synonym: Murine Plus,Tetryzoline hydrochloride,Tyzine,Tetrahydrozoline HCl
Target: Adrenergic Receptor
2-BFI hydrochloride
T22492
Synonym:
Target: Imidazoline Receptor
Rilmenidine hemifumarate
T21911
Synonym: Rilmenidine (hemifumarate),S-3341 hemifumarate
Target: Apoptosis, Imidazoline Receptor
RS 45041-190 hydrochloride
T23263
Synonym:
Target: Others
Efaroxan hydrochloride
T22760
Synonym:
Target: Others
S23757
T26171
Synonym: S-23757,S 23757
Target:
Tracizoline
T68931
Synonym:
Target:
Moxonidine hydrochloride
T40869
Synonym: BDF5895hydrochloride
Target:
Dexisometheptene
T27155
Synonym: TNX 201,TNX-201,(R)-Isometheptene,TNX201
Target:
RX 801077
T73214
Synonym: 2 BFI free base
Target:
1 2
TargetMol