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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T22051 | BU 224 hydrochloride | Imidazoline Receptor | |
BU 224 hydrochloride is a selective imidazoline I(2) binding site ligand and has antinociceptive and antidepressant-like activities. | |||
T6641 | Rilmenidine Phosphate | Apoptosis , Adrenergic Receptor , Autophagy , Imidazoline Receptor | |
Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension. | |||
T3158 | Harmane | Loturine,Harman,Aribine | Adrenergic Receptor , Monoamine Oxidase , Imidazoline Receptor |
Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke. | |||
T0115 | Idazoxan hydrochloride | RX 781094 | Adrenergic Receptor , Imidazoline Receptor |
Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity. | |||
T0925 | Allantoin | Glyoxyldiureide,5-Ureidohydantoin | Endogenous Metabolite , Imidazoline Receptor |
Allantoin (Glyoxyldiureide), a urea hydantoin found in urine and plants, is used in dermatological preparations. | |||
T22052 | BU 226 hydrochloride | Imidazoline Receptor | |
BU 226 hydrochloride demonstrates affinity for imidazoline (I) receptors, in particular the I2 binding site with a Ki of 1.4 nM. BU 226 hydrochloride showed low (microM) affinity for alpha 2-adrenoceptors. | |||
T1028 | Moxonidine | BDF5895 | Imidazoline Receptor |
Moxonidine (BDF5895) is a selective agonist at the imidazoline receptor subtype 1, acting as an antihypertensive drug. | |||
T4808 | Agmatine sulfate | Agmatine sulfate salt | Endogenous Metabolite , NO Synthase , Imidazoline Receptor |
Agmatine sulfate (Agmatine sulfate salt) is a bioactive metabolite of the arginine amino acid. It exerts modulatory action at multiple molecular targets, such as neurotransmitter systems, ion channels and nitric oxide sy... | |||
T23283 | 2-Methoxyidazoxan monohydrochloride | RX 821002 hydrochloride | Adrenergic Receptor |
L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor, with little or no antagonistic effect on imidazoline. It has a significantly higher affinity ... | |||
T15010 | CR4056 | 6-(1H-imidazol-1-yl)-2-phenylquinazoline | MAO , Imidazoline Receptor |
CR4056 (6-(1H-imidazol-1-yl)-2-phenylquinazoline) is a selective inhibitor of MAO-A with IC50 of 202.7 nM and a ligand of I2-imidazoline receptor with IC50 of 596 nM. | |||
T6703 | Tetrahydrozoline hydrochloride | Murine Plus,Tetryzoline hydrochloride,Tyzine,Tetrahydrozoline HCl | Adrenergic Receptor |
Tetrahydrozoline hydrochloride (Murine Plus) is an imidazoline derivative with alpha receptor agonist activity. | |||
T22492 | 2-BFI hydrochloride | Imidazoline Receptor | |
2-BFI hydrochloride is a high-affinity agonist of I2-imidazoline receptor. 2-BFI hydrochloride can be used in studies about protection against stroke and acute inflammatory immune disease. | |||
T21911 | Rilmenidine hemifumarate | Rilmenidine (hemifumarate),S-3341 hemifumarate | Apoptosis , Imidazoline Receptor |
Rilmenidine hemifumarate (S-3341 hemifumarate) is a novel, orally active and selective I1 imidazoline receptor and α2-adrenoceptor agonist that induces autophagy, regulates the proliferation of leukaemia cells, stimulate... | |||
T23263 | RS 45041-190 hydrochloride | Others | |
Highly selective I2 imidazoline receptor ligand | |||
T22760 | Efaroxan hydrochloride | Others | |
α2 adrenoceptor antagonist and imidazoline I1 receptor ligand | |||
T26171 | S23757 | S-23757,S 23757 | |
S23757 is an imidazoline 1 receptor (I1R) selective ligand. | |||
T68931 | Tracizoline | ||
Tracizoline is a potent I2-imidazoline receptor agonist. | |||
T40869 | Moxonidine hydrochloride | BDF5895hydrochloride | |
Moxonidine Hydrochloride serves as a selective agonist for the imidazoline receptor subtype 1 and functions as an antihypertensive agent. It primarily acts within the central nervous system and demonstrates a significant... | |||
T27155 | Dexisometheptene | TNX 201,TNX-201,(R)-Isometheptene,TNX201 | |
Dexisometheptene is an antimigraine drug candidate. Dexisometheptene significantly increases the pain threshold of acute pain response, and potently and selectively binds to receptors in the central nervous system known ... | |||
T73214 | RX 801077 | 2 BFI free base | |
RX 801077 (2 BFI free base), a selective imidazoline I2 receptor (I2R) agonist, exhibits a K i value of 70.1 nM, demonstrating anti-inflammatory and neuroprotective properties. This compound holds research potential for ... |